U-69593

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Opioid receptor ligand

Selective κ-opioid agonist. Thought to be selective for the κ-1 subtype (K_D=3.8nM in human cerebral cortex membranes). Immunomodulatory activity.

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Appearance	White solid.
CAS	96744-75-1
Couple Target	Opioid receptor
Couple Type	Ligand
Formula	C₂₂H₃₂N₂O₂
MW	356.5
Purity	≥99% (TLC)
Solubility	Soluble in 100% ethanol, 0.1N hydrogen chloride, or DMSO. Insoluble in water or 0.1N sodium hydroxide.
Source	Synthetic.

Use/Stability	As indicated on product label or CoA when stored as recommended. Store, as supplied, -20°C for up to 1 year. Store solutions at -20°C for up to 3 months.
Long Term Storage	-20°C
Shipping	Ambient Temperature

Regulatory Status	RUO – Research Use Only

Ligand binding profiles of U-69, 593-sensitive and-insensitive sites in human cerebral cortex membranes: evidence of kappa opioid receptors heterogeneity: K.W. Kim et al.; Life Sci. 58, 1671 (1996), Abstract
Immunomodulatory activity of mu- and kappa-selective opioid agonists: D.D. Taub et al.; PNAS 88, 360 (1991), Abstract
Kappa-opioid receptors and analgesia: M.J. Millan; Trends Pharmacol. Sci. 11, 70 (1990), Abstract
Pharmacological activities of optically pure enantiomers of the kappa opioid agonist, U50,488, and its cis diastereomer: evidence for three kappa receptor subtypes: R.B. Rothman et al.; Eur. J. Pharmacol. 167, 345 (1989), Abstract

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