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KT5720

BML-EI199

12 citations

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PKA inhibitor

KT5720 is a hexylester derivative of K-252a and is a selective inhibitor of PKA (K_i=0.056 µM). Cell permeable.

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Product Details

Appearance	White powder.
CAS	108068-98-0
Couple Target	PKA
Couple Type	Inhibitor
Formula	C₃₂H₃₁N₃O₅
MW	537.6
Purity	≥98% (HPLC)
Solubility	Soluble in methanol: clear colorless solution at 5mg/ml.

Handling & Storage

Use/Stability	As indicated on product label or CoA when stored as recommended. Stable for at least 1 year after receipt when stored, as supplied, at -20°C. Stock solutions are stable for up to 3 months at -20°C.
Handling	Protect from light.
Long Term Storage	-20°C
Shipping	Ambient Temperature

Regulatory Status	RUO – Research Use Only

Phosphorylation of the compartmentalized PKA substrate TAF15 regulates RNA-protein interactions: Feichtner, A., Enzler, F., et al.; Cell. Mol. Life Sci. 81, 162 (2024), Abstract
Laminin 211 inhibits protein kinase A in Schwann cells to modulate neuregulin 1 type III-driven myelination: Ghidinelli, M., Poitelon, Y., et al.; PLoS Biol. 15, e2001408 (2017), Abstract
Olig2-Targeted G-Protein-Coupled Receptor Gpr17 Regulates Oligodendrocyte Survival in Response to Lysolecithin-Induced Demyelination: Ou, Z., Sun, Y., et al.; J. Neurosci. 36, 10560 (2016), Abstract
Adrenergic and serotonin receptors affect retinal superoxide generation in diabetic mice: relationship to capillary degeneration and permeability: Du, Y., Cramer, M., et al.; FASEB J. 29, 2194 (2015), Abstract
Cilostazol Upregulates Autophagy via SIRT1 Activation: Reducing Amyloid-β Peptide and APP-CTFβ Levels in Neuronal Cells: Lee, H. R., Shin, H. K., et al.; PLoS One 10, e0134486 (2015), Abstract
Dissociations in the effects of β2-adrenergic receptor agonists on cAMP formation and superoxide production in human neutrophils: support for the concept of functional selectivity: Brunskole Hummel, I., Reinartz, M. T., et al.; PLoS One 8, e64556 (2013), Abstract
Evidence for a novel anti-apoptotic pathway in human keratinocytes involving the aryl hydrocarbon receptor, E2F1, and checkpoint kinase 1: Frauenstein, K., Sydlik, U., et al.; Cell Death Differ. 20, 1425 (2013), Abstract
Protein kinase A phosphorylation activates Vpr-induced cell cycle arrest during human immunodeficiency virus type 1 infection: Barnitz, R. A., Wan, F., et al.; J. Virol. 84, 6410 (2010), Abstract
Effects of insulin, insulin-like growth factor-I, and phorbol esters on neutral cholesteryl esterase activity in cultured rat vascular smooth muscle cells.: R. Fujiwara, et al.; J. Lab. Clin. Med. 126, 240 (1995), Abstract
Effects of selective inhibition of protein kinase C, cyclic AMP-dependent protein kinase, and Ca(2+)-calmodulin-dependent protein kinase on neurite development in cultured rat hippocampal neurons: L. Cabell & G. Audesirk; Int. J. Dev. Neurosci. 11, 357 (1993), Abstract

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KT5720

BML-EI199

Product Details

Handling & Storage

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