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ET_A receptor antagonist [BQ-123] . sodium salt

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Highly potent and selective ET_Aantagonist.

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CAS	136553-81-6
Formula	C₃₁H₄₂N₆O₇ . Na
MW	633.7
Purity	≥96%
Quantity	*Sold as net peptide weight.
Sequence	cyclo(D-Asp-Pro-D-Val-Leu-D-Trp . Na)
Solubility	Soluble in water.

Use/Stability	As indicated on product label or CoA when stored as recommended. Stable for at least 3 years after receipt when stored at -20°C. Stock solutions are stable for up to 3 months when stored at -20°C.
Long Term Storage	-20°C
Shipping	Ambient Temperature

Regulatory Status	RUO – Research Use Only

Endothelin: progress in pharmacology and physiology: W.G. Haynes, et al.; TIPS 14, 225 (1993), (Review), Abstract
Biological profiles of highly potent novel endothelin antagonists selective for the ETA receptor: M. Ihara, et al.; Life Sci. 50, 247 (1992), Abstract
Conformational study of cyclo[D-Trp-D-Asp-Pro-D-Val-Leu], an endothelin- A receptor-selective antagonist: R.A. Atkinson & J.T. Pelton; FEBS Lett. 296, 1 (1992), Abstract
A novel ETA antagonist (BQ-123) inhibits endothelin-1-induced phosphoinositide breakdown and DNA synthesis in rat vascular smooth muscle cells: S. Eguchi, et al.; FEBS Lett. 302, 243 (1992), Abstract
Identification of a domain of ETA receptor required for ligand binding: M. Adachi, et al.; FEBS Lett. 311, 179 (1992), Abstract
Cyclic pentapeptide endothelin antagonists with high ETA selectivity. Potency- and solubility-enhancing modifications: K. Ishikawa, et al.; J. Med. Chem. 35, 2139 (1992), Abstract

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