AM-630

BML-CR107

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Cannabinoid receptor ligand

Acts as a cannabinoid receptor antagonist in mouse brain, vas deferens and guinea pig brain, but an agonist in guinea pig ileum. Acts as an inverse agonist on cloned human CB₁ receptors.

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Product Details

Appearance	White to off-white solid.
CAS	164178-33-0
Couple Target	Cannabinoid receptor
Couple Type	Ligand
Formula	C₂₃H₂₅IN₂O₃
MW	504.4
Purity	≥98% (TLC)
Solubility	Soluble in DMSO or dimethyl formamide.

Handling & Storage

Use/Stability	As indicated on product label or CoA when stored as recommended.
Handling	Store under inert gas and avoid exposure to light.
Long Term Storage	-20°C
Shipping	Ambient Temperature

Regulatory Status	RUO – Research Use Only

Activation of murine microglial N9 cells is attenuated through cannabinoid receptor CB2 signaling: L. Ma, et al.; Biochem. Biophys. Res. Commun. 458, 92 (2015), Application(s): Cell Culture, Abstract
Endogenous anandamide and cannabinoid receptor-2 contribute to electroacupuncture analgesia in rats: Chen, L., Zhang, J., et al.; J. Pain 10, 732 (2009), Abstract
Effects of the cannabinoid antagonists AM281 and AM630 on deprivation-induced intake in Lewis rats: N.A. Werner & J.E. Koch; Brain Res. 967, 290 (2003), Abstract
Agonist-inverse agonist characterization at CB1 and CB2 cannabinoid receptors of L759633, L759656, and AM630: R.A. Ross et al.; Br. J. Pharmacol. 126, 665 (1999), Abstract
AM630 is an inverse agonist at the human cannabinoid CB1 receptor: R.S. Landsman et al.; Life Sci. 62, PL109 (1998), Abstract
AM630 is a competitive cannabinoid receptor antagonist in the guinea pig brain: K. Hosohata et al.; Life Sci. 61, PL115 (1997), Abstract
AM630, a competitive cannabinoid receptor antagonist: R. Pertwee et al.; Life Sci 56, 1949 (1995), Abstract

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AM-630

BML-CR107

Product Details

Handling & Storage

Datasheet, Manuals, SDS & CofA

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