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A1874

ENZ-CHM262

  • ENZ-CHM262-0005   —   5 mg
    $1,047.00
  • ENZ-CHM262-0010   —   10 mg
    $1,460.00
  • ENZ-CHM262-0025   —   25 mg
    $2,996.00

A1874 is a nutlin-based PROTAC targeting on BRD4, consist of a BRD4-ligand JQ1 linked to a MDM2 E3 ligase ligand RG7388. A1874 possesses dual function as it dose-dependently degraded its target BRD4, accompanied with the downregulation of c-MYC, as well as stabilization of P53 and upregulated P21 due to the efficient engagement of MDM2 by RG7388.

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Regulatory Status

RUO – Research Use Only